Affiliations 

  • 1 Department of Chemistry, School of Advanced Sciences, Vellore Institute of Technology, Vellore-632014, Tamil Nadu, India
  • 2 VIT School of Agricultural Innovations and Advanced Learning, Vellore Institute of Technology, Vellore- 632014, Tamil Nadu, India
  • 3 School of Pharmacy, Suresh Gyan Vihar University, Jagatpura-302017, Mahal Road, Jaipur, India
  • 4 Department of Life Sciences, School of Pharmacy, International Medical University, 57000 Bukit Jalil, Kuala Lumpur, Malaysia
  • 5 Pharmaceutical Chemistry Unit, Faculty of Pharmacy, AIMST University, Bedong, Kedah, Darul, Aman, Malaysia
  • 6 School of Pharmaceutical Sciences, Lovely Professional University, Phagwara- 144411, Punjab, India
  • 7 Discipline of Pharmacy, Graduate School of Health, University of Technology Sydney (UTS), Ultimo, NSW, 2007, Australia
PMID: 33573582 DOI: 10.2174/1871523020666210126144506

Abstract

AIMS: The present investigation was aimed at exploring the phytoconstituents using Gas Chromatography Mass Spectroscopy and to evaluate antioxidant and anti-inflammatory properties of the leaf extracts.

MATERIALS AND METHODS: The extracts were obtained sequentially with petroleum ether, ethyl acetate and water using Soxhlet apparatus. The anti-inflammatory property of the identified compounds using GC- MS spectroscopy was evaluated in silico. The antioxidant activity was performed by DPPH and H2O2 method whereas anti-inflammatory study was carried out by HRBC membrane stabilization method. Terpenoids were found to be a major constituents in petroleum ether extract while, phenols and flavonoids were predominantly found in ethyl acetate extract.

RESULTS AND DISCUSSION: The GC-MS analysis of the extract revealed six major molecules including Squalene, 19β, 28-epoxyleanan-3-ol and 2-tu-Butyl-5-chloromethyl-3-methyl-4-oxoimidazolidine- 1-carboxylic acid. The ethyl acetate extract showed a significant antioxidant activity (P<0.01) in both DPPH method (70.87%) and H2O2 method (73.58%) at 200 μg mL-1. Increased membrane stabilization of petroleum ether extract was observed in the in vitro anti-inflammatory activity study. A strong relationship between the terpenoid content and anti-inflammatory activity was obtained from the correlation (0.971) and docking study.

CONCLUSION: These results justify T. involucrata to be a rich source of terpenoids with potent anti- inflammatory property.

* Title and MeSH Headings from MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine.